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SB756050
SKU
HY-102016-10 mg
Category Reference compound
Tags G protein-coupled Bile Acid Receptor 1, GPCR/G Protein, Metabolic Disease
$50 – $180
Products Details
Product Description
– SB756050 is a selective TGR5 agonist. SB756050 has the potential for type 2 diabetes treatment.
Web ID
– HY-102016
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Metabolism-sugar/lipid metabolism
Molecular Formula
– C21H28N2O8S2
References
– [1]Hodge RJ, et al. Safety, Pharmacokinetics, and Pharmacodynamic Effects of a Selective TGR5 Agonist, SB-756050, in Type 2 Diabetes. Clin Pharmacol Drug Dev. 2013 Jul;2(3):213-22.
CAS Number
– 447410-57-3
Molecular Weight
– 500.59
Compound Purity
– 98.49
SMILES
– O=S(N1CCN(S(=O)(C2=CC=C(OC)C(OC)=C2)=O)CCC1)(C3=CC=C(OC)C(OC)=C3)=O
Clinical Information
– Phase 1
Research Area
– Metabolic Disease
Solubility
– DMSO : ≥ 150 mg/mL
Target
– G protein-coupled Bile Acid Receptor 1
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.