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S1P2 antagonist 1
Products Details
Product Description
– S1P2 antagonist 1 is an orally bioavailable S1P2 antagonist against fibrotic diseases.
Web ID
– HY-141845
Shipping
– Room temperature
Applications
– Neuroscience-Neuromodulation
Molecular Formula
– C23H21ClN4O4
References
– [1]Mammoliti O, et al. Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases. J Med Chem. 2021 Oct 14;64(19):14557-14586.
CAS Number
– 2262402-83-3
Molecular Weight
– 452.89
SMILES
– OC([C@@H](C)N1N=C(CN2N=C(C=C(Cl)C(OCC3CC3)=C4)C4=C2)C5=CC=CC=C5C1=O)=O
Clinical Information
– No Development Reported
Research Area
– Others
Solubility
– 10 mM in DMSO
Target
– LPL Receptor
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.