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Products Details
Product Description
– (S)-BI-1001 (Compound 11) is an active S-enantiomer of BI-1001. (S)-BI-1001 exhibits antiviral potency against HIV-1 integrase with an IC50 of 28 nM, an EC50 of 450 nM and a Kd of 4.7 μM[1].
Web ID
– HY-12210
Shipping
– Room temperature
Applications
– COVID-19-anti-virus
Molecular Formula
– C19H15BrClNO3
References
– [1]Fader LD, et al. Discovery of BI 224436, a Noncatalytic Site Integrase Inhibitor (NCINI) of HIV-1. ACS Med Chem Lett. 2014 Jan 22;5(4):422-7.
CAS Number
– 957889-73-5
Molecular Weight
– 420.68
SMILES
– ClC1=CC=C(C2=C(C=C(Br)C=C3)C3=NC(C)=C2[C@H](OC)C(O)=O)C=C1
Clinical Information
– No Development Reported
Research Area
– Infection
Solubility
– 10 mM in DMSO
Target
– HIV Integrase
Pathway
– Metabolic Enzyme/Protease
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
