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PSB11 (hydrochloride)
Products Details
Product Description
– PSB11 hydrochloride is an antagonist with reverse excitatory activity for human A3 Adenosine Receptor with high affinity (Ki=2.3 nM)[1].
Web ID
– HY-103176
Shipping
– Room temperature
Molecular Formula
– C16H18ClN5O
References
– [1]Müller C E, et al. [3H] 8-Ethyl-4-methyl-2-phenyl-(8R)-4, 5, 7, 8-tetrahydro-1H-imidazo [2, 1-i]-purin-5-one ([3H] PSB-11), a novel high-affinity antagonist radioligand for human A3 adenosine receptors[J]. Bioorganic & medicinal chemistry letters, 2002, 12(3): 501-503.
CAS Number
– 453591-58-7
Molecular Weight
– 331.80
SMILES
– O=C1N(C)C2=C(N=C(C3=CC=CC=C3)N2)C4=N[C@H](CC)CN14.[H]Cl
Clinical Information
– No Development Reported
Research Area
– Others
Solubility
– 10 mM in DMSO
Target
– Adenosine Receptor
Isoform
– Adenosine A3 receptor (A3R)
Pathway
– GPCR/G Protein
Product type
– Reference compound
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