Pirenperone

$45$460

Products Details

Product Description

– Pirenperone (R 47465) is a 5-HT2 serotonin receptor antagonist. Pirenperone exhibits modest anxiolytic activity[1][2].

Web ID

– HY-B1737

Storage Temperature

– -20°C, 3 years; 4°C, 2 years (Powder)

Shipping

– Room Temperature

Applications

– Neuroscience-Neuromodulation

Molecular Formula

– C23H24FN3O2

References

– [1]Krstić MK, et, al. Divergent effects of pirenperone, a 5-HT2 antagonist, on the pressor and tachycardic responses to 5-HT in guinea-pigs. Arch Int Physiol Biochim. 1983 Nov;91(4):345-9. |[2]Ansseau M, et, al. Pilot study of a specific serotonergic antagonist, pirenperone, in the treatment of anxiety disorders. Acta Psychiatr Belg. Sep-Oct 1983;83(5):517-24.

CAS Number

– 75444-65-4

Molecular Weight

– 393.45

Compound Purity

– 98.74

SMILES

– O=C1C(CCN2CCC(C(C3=CC=C(F)C=C3)=O)CC2)=C(C)N=C4N1C=CC=C4

Clinical Information

– No Development Reported

Research Area

– Neurological Disease

Solubility

– 0.1 M HCL : 16.67 mg/mL (ultrasonic;warming;adjust pH to 3 with 0.1 M HCL;heat to 60°C)|DMSO : 25 mg/mL (ultrasonic;warming;heat to 60°C)

Target

– 5-HT Receptor

Pathway

– GPCR/G Protein;Neuronal Signaling

Product type

– Reference compound

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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