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Products Details
Product Description
– Piprofurol is a calcium channel inhibitor. Piprofurol inhibites in a concentration-dependent manner the calcium-induced contractions in isolated potassium depolarized preparations of rat aorta and relaxes the K+-induced contraction of the dog coronary artery and the rabbit basilar artery. Piprofurol exerts a negative inotropic effect on guinea-pig papillary muscle, with the EC50 of 5 μM[1].
Web ID
– HY-114920
Shipping
– Room temperature
Molecular Formula
– C26H33NO6
References
– [1]Pourrias B, et al. Calcium blocking properties of piprofurol. Arch Int Pharmacodyn Ther. 1985;274(2):223-239.
CAS Number
– 40680-87-3
Molecular Weight
– 455.54
SMILES
– OC(C1=C(C(OC)=C2OC=CC2=C1OC)OCCN3CCCCC3)CCC4=CC=C(C=C4)O
Clinical Information
– No Development Reported
Research Area
– Cardiovascular Disease
Solubility
– 10 mM in DMSO
Target
– Calcium Channel
Pathway
– Membrane Transporter/Ion Channel;Neuronal Signaling
Product type
– Reference compound
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