Download Files:
Piperidine-GNE-049-N-Boc
SKU
HY-134592-10 mg
Category Reference compound
Tags Cancer, Ligands for Target Protein for PROTAC, PROTAC
$950 – $8,600
Products Details
Product Description
– Piperidine-GNE-049-N-Boc is a ligand for target protein for PROTAC of dCBP-1 (HY-134582). dCBP-1 is a potent and selective heterobifunctional degrader of p300/CBP[1].
Web ID
– HY-134592
Storage Temperature
– 4°C (Powder, sealed storage, away from moisture and light)
Shipping
– Room Temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C30H39F2N7O2
References
– [1]Vannam R, et, al. Targeted degradation of the enhancer lysine acetyltransferases CBP and p300. Cell Chem Biol. 2020 Dec 31;S2451-9456(20)30513-4.
CAS Number
– 1936431-36-5
Molecular Weight
– 567.67
Compound Purity
– 98.82
SMILES
– O=C(N1CCC(N(C2CCNCC2)N=C3N4CCCC5=C4C=C(C(F)F)C(C6=CN(C)N=C6)=C5)=C3C1)OC(C)(C)C
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 1M HCl : 32.5 mg/mL (ultrasonic;adjust pH to 1 with HCl)
Target
– Ligands for Target Protein for PROTAC
Pathway
– PROTAC
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.