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PD-168077 maleate
$100 – $880
Products Details
Product Description
– PD-168077 maleate is a selective dopamine D4 receptor agonist, with a Ki of 9 nM.
Web ID
– HY-21098A
Storage Temperature
– 4°C (Powder, sealed storage, away from moisture)
Shipping
– Room Temperature
Applications
– Neuroscience-Neuromodulation
Molecular Formula
– C24H26N4O5
References
– [1]Clifford JJ, et al. Topographically based search for an “Ethogram” among a series of novel D(4) dopamine receptor agonists and antagonists. Neuropsychopharmacology. 2000 May;22(5):538-44.|[2]Gu Z, et al. Activation of dopamine D4 receptors induces synaptic translocation of Ca2+/calmodulin-dependent protein kinase II in cultured prefrontal cortical neurons. Mol Pharmacol. 2006 Mar;69(3):813-22.
CAS Number
– 630117-19-0
Molecular Weight
– 450.49
Compound Purity
– 98.74
SMILES
– O=C(NCN1CCN(C2=CC=CC=C2C#N)CC1)C3=CC=CC(C)=C3.O=C(O)/C=CC(O)=O
Clinical Information
– No Development Reported
Research Area
– Neurological Disease
Solubility
– DMSO : 150 mg/mL (ultrasonic)|H2O : ≥ 0.1 mg/mL
Target
– Dopamine Receptor
Isoform
– D4 Receptor
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
