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Products Details
Product Description
– PCSK9-IN-22 (compound 29) is an orally active inhibitor of PCSK9. PCSK9-IN-22 inhibits the interaction of the protein with LDLR in vivo[1].
Web ID
– HY-160036
Shipping
– Room temperature
Molecular Formula
– C28H30N6O
References
– [1]Phillip Albert Coghlan, et al. Heterocyclic inhibitors of pcsk9. WO2022133529A1. 2022-06-30.
CAS Number
– 2794203-47-5
Molecular Weight
– 466.58
SMILES
– N[C@@H](CCC1)CN1CC2=CC(NC(C3=CC(C4=CC=CC=C4)=CC=N3)=O)=CC(N5C=NC(C)=C5)=C2
Clinical Information
– No Development Reported
Research Area
– Metabolic Disease
Solubility
– 10 mM in DMSO
Target
– Ser/Thr Protease
Pathway
– Metabolic Enzyme/Protease
Product type
– Reference compound
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