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PBRM1-BD2-IN-3
$315
Only 1000 item(s) left in stock.
Products Details
Product Description
– PBRM1-BD2-IN-3 (compound 12) is a potent PBRM1-BD2 inhibitor with an IC50 value of 1.1 μM. PBRM1-BD2 Inhibitor can be used to research anticancer[1].
Web ID
– HY-151530
Shipping
– Room temperature
Molecular Formula
– C14H11ClN2O
References
– [1]Shishodia S, et al. Selective and Cell-Active PBRM1 Bromodomain Inhibitors Discovered through NMR Fragment Screening. J Med Chem. 2022 Oct 13.
CAS Number
– 2819989-58-5
Molecular Weight
– 258.70
SMILES
– O=C1NC(C2=CC=CC=C2)NC3=C1C(Cl)=CC=C3
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Epigenetic Reader Domain
Pathway
– Epigenetics
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.