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Products Details
Product Description
– NSC 698600 is a potent PCAF inhibitor, with IC50 of 6.51 µM (PCAF/H31-21). NSC 698600 exhibits good activity of inhibiting the proliferation of cancer cells[1].
Web ID
– HY-147289
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C14H12N2O2S
References
– [1]Furdas SD, et al. Synthesis and biological testing of novel pyridoisothiazolones as histone acetyltransferase inhibitors. Bioorg Med Chem. 2011 Jun 15;19(12):3678-89.
CAS Number
– 908069-17-0
Molecular Weight
– 272.32
SMILES
– O=C1C2=CC(C)=CN=C2SN1C3=CC=C(C=C3)OC
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Histone Acetyltransferase
Isoform
– GCN5/PCAF
Pathway
– Epigenetics
Product type
– Reference compound
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