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NCRW0005-F05
$85 – $780
Products Details
Product Description
– NCRW0005-F05 is a potent GPR139 antagonist with an IC50 value of 0.21 μM. NCRW0005-F05 can be used to research diabetes, obesity and Parkinson’s disease[1].
Web ID
– HY-128057
Storage Temperature
– -20°C, 3 years (Powder)
Shipping
– Blue Ice
Applications
– Metabolism-protein/nucleotide metabolism
Molecular Formula
– C16H13F2NO2
References
– [1]Wang J, et al. High-throughput screening of antagonists for the orphan G-protein coupled receptor GPR139. Acta Pharmacol Sin. 2015 Jul;36(7):874-8.
CAS Number
– 342779-66-2
Molecular Weight
– 289.28
Compound Purity
– 99.0
SMILES
– O=C1N(C2=CC=CC=C2)C(C3=CC=C(OC)C=C3)C1(F)F
Clinical Information
– No Development Reported
Research Area
– Metabolic Disease; Neurological Disease
Solubility
– DMSO : ≥ 100 mg/mL
Target
– GPR139
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
