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Products Details
Product Description
– MRS2298? is a potent acyclic P2Y1 receptor antagonist with a Ki of 29.6 nM. MRS2298 inhibits the ADP-induced aggregation of human platelets with an IC50 of 62.8 nM. MRS2298 inhibits Ca2+ rise in platelets with an IC50 of 810 nM[1].
Web ID
– HY-113723
Shipping
– Room temperature
Molecular Formula
– C10H16ClN5O8P2
References
– [1]Marco Cattaneo, et al. Antiaggregatory activity in human platelets of potent antagonists of the P2Y 1 receptor. Biochem Pharmacol. 2004 Nov 15;68(10):1995-2002.
CAS Number
– 491611-43-9
Molecular Weight
– 431.66
SMILES
– O=P(OCC(COP(O)(O)=O)CN1C=NC2=C(N=C(N=C12)Cl)NC)(O)O
Clinical Information
– No Development Reported
Research Area
– Cardiovascular Disease
Solubility
– 10 mM in DMSO
Target
– P2Y Receptor
Pathway
– GPCR/G Protein
Product type
– Reference compound
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