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MRS1186
SKU
HY-118678-Get quote
Category Reference compound
Tags Adenosine Receptor, GPCR/G Protein, Inflammation/Immunology
Products Details
Product Description
– MRS1186 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM.
Web ID
– HY-118678
Shipping
– Room temperature
Applications
– COVID-19-immunoregulation
Molecular Formula
– C16H12ClN5O2
References
– [1]Tafi A, et al. Pharmacophore based receptor modeling: the case of adenosine A3 receptor antagonists. An approach to the optimization of protein models. J Med Chem. 2006 Jul 13;49(14):4085-97.
CAS Number
– 183721-03-1
Molecular Weight
– 341.75
SMILES
– CCC(NC1=NC2=C(C3=NC(C4=CC=CO4)=NN13)C=C(C=C2)Cl)=O
Clinical Information
– No Development Reported
Research Area
– Inflammation/Immunology
Solubility
– 10 mM in DMSO
Target
– Adenosine Receptor
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.