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MM 07
$190 – $1,338
Products Details
Product Description
– MM 07 is a biased apelin receptor agonist, with a KD of 300 nM in CHO-K1 cells and a KD of 172 nM in human heart.
Web ID
– HY-108003
Storage Temperature
– -80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture)
Shipping
– Blue Ice
Applications
– COVID-19-immunoregulation
Molecular Formula
– C67H106N22O14S3
References
– [1]Brame AL, et al. Design, characterization, and first-in-human study of the vascular actions of a novel biased apelin receptor agonist. Hypertension. 2015 Apr;65(4):834-40.
CAS Number
– 1876450-21-3
Molecular Weight
– 1539.89
Compound Purity
– 98.08
SMILES
– O=C([C@H]1N(CCC1)C(CNC([C@H](CCCCN)NC([C@@H](NC([C@H]2NC([C@](NC([C@@H](NC([C@@]3([H])N(CCC3)C([C@@](CCCNC(N)=N)([H])NC([C@@H](N)CSSC2)=O)=O)=O)CCCNC(N)=N)=O)([H])CC(C)C)=O)=O)CC4=CN=CN4)=O)=O)=O)N[C@@H](CCSC)C(N5[C@@H](CCC5)C(N[C@H](C(O)=O)CC6=CC=CC=C6)=O)=O
Clinical Information
– No Development Reported
Research Area
– Cardiovascular Disease
Solubility
– DMSO : 62.5 mg/mL (ultrasonic)
Target
– Apelin Receptor (APJ)
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
