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MEK4 inhibitor-2
Products Details
Product Description
– MEK4 inhibitor-2 is a novel MEK4 inhibitor against pancreatic adenocarcinoma with an IC50 value of 83 nM.
Web ID
– HY-139639
Shipping
– Room temperature
Applications
– Cancer-Kinase/protease
Molecular Formula
– C20H15FN4O3S
References
– [1]Kwong AJ, et al. Rational Design, Optimization, and Biological Evaluation of Novel MEK4 Inhibitors against Pancreatic Adenocarcinoma. ACS Med Chem Lett. 2021 Sep 15;12(10):1559-1567.
CAS Number
– 2833643-78-8
Molecular Weight
– 410.42
SMILES
– FC1=CC=C(C(C2=CC=CC(S(=O)(NC3=CC=C(C(N)=O)C=C3)=O)=C2)=NN4)C4=C1
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– MEK
Pathway
– MAPK/ERK Pathway
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.