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LPA2 antagonist 1
$350 – $2,100
Products Details
Product Description
– LPA2 antagonist 1 is a LPA2 antagonist with an IC50 of 17 nM.
Web ID
– HY-18075
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Cancer-Kinase/protease
Molecular Formula
– C20H23Cl2N5O2S2
References
– [1]Beck HP, et al. Discovery of potent LPA2 (EDG4) antagonists as potential anticancer agents. Bioorg Med Chem Lett. 2008 Feb 1;18(3):1037-41.
CAS Number
– 1017606-66-4
Molecular Weight
– 500.46
Compound Purity
– 99.56
SMILES
– ClC1=C(Cl)C=C(S(=O)(N2CCN(C[C@@H](NC3=NC=NC4=C3SC=C4C)C)CC2)=O)C=C1
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– DMF : ≥ 100 mg/mL|DMSO : ≥ 100 mg/mL
Target
– LPL Receptor
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
