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Lavoltidine
SKU
HY-121450-Get quote
Category Reference compound
Tags Cancer, GPCR/G Protein;Immunology/Inflammation;Neuronal Signaling, Histamine Receptor
Products Details
Product Description
– Lavoltidine (Loxtidine) is an an orally active, irreversible and highly potent histamine H2-receptor antagonist. Lavoltidine strongly inhibits gastric acid secretion and also induces hypergastrinemia[1].
Web ID
– HY-121450
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C19H29N5O2
References
– [1]Takaishi S, et al. Synergistic inhibitory effects of gastrin and histamine receptor antagonists on Helicobacter-induced gastric cancer.
CAS Number
– 76956-02-0
Molecular Weight
– 359.47
SMILES
– OCC1=NN(C(NCCCOC2=CC=CC(CN3CCCCC3)=C2)=N1)C
Clinical Information
– Phase 2
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Histamine Receptor
Isoform
– H2 Receptor
Pathway
– GPCR/G Protein;Immunology/Inflammation;Neuronal Signaling
Product type
– Reference compound
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