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hGPR91 antagonist 3
$400 – $1,350
Products Details
Product Description
– hGPR91 antagonist 3 (Compound 5g) is a potent and orally active GPR91 antagonist with IC50 of 35 nM and 135 nM, for human GPR91 and rat GPR91, respectively[1].
Web ID
– HY-145919
Storage Temperature
– 4°C (Powder, stored under nitrogen)
Shipping
– Room Temperature
Applications
– COVID-19-immunoregulation
Molecular Formula
– C23H18F4N4O2
References
– [1]Bhuniya D, et al. Discovery of a potent and selective small molecule hGPR91 antagonist. Bioorg Med Chem Lett. 2011;21(12):3596-3602.
CAS Number
– 1314796-31-0
Molecular Weight
– 458.41
Compound Purity
– 98.82
SMILES
– O=C(CCCC1=CC=C2C=CC=NC2=N1)NCC3=CC(C4=CC(C(F)(F)F)=C(F)C=C4)=NO3
Clinical Information
– No Development Reported
Research Area
– Inflammation/Immunology; Cardiovascular Disease
Solubility
– 10 mM in DMSO
Target
– Succinate Receptor 1
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
