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hGPR91 antagonist 1
$260 – $2,100
Products Details
Product Description
– hGPR91 antagonist 1 (Compound 4c) is a potent and selective GPR91 antagonist with an IC50 of 7 nM for human GPR91[1].
Web ID
– HY-126217
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Metabolism-protein/nucleotide metabolism
Molecular Formula
– C31H23F4N3O
References
– [1]Bhuniya D, et al. Discovery of a potent and selective small molecule hGPR91 antagonist. Bioorg Med Chem Lett. 2011 Jun 15;21(12):3596-602.
CAS Number
– 1314796-00-3
Molecular Weight
– 529.53
Compound Purity
– 98.71
SMILES
– O=C(N[C@@H](C)C1=CC=C(C2=CC=C(F)C(C(F)(F)F)=C2)C=C1)CC3=CC=C(C4=NC5=NC=CC=C5C=C4)C=C3
Clinical Information
– No Development Reported
Research Area
– Metabolic Disease
Solubility
– DMSO : ≥ 125 mg/mL
Target
– Succinate Receptor 1
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
