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GST-IN-1

Products Details

Product Description

– GST-IN-1 (compound 16) is a glutathione S-transferase (GST) inhibitor with IC50s of 1.55 μM (sjGST) and 2.02 μM (hGSTM2), respectively.

Web ID

– HY-149419

Shipping

– Room temperature

Molecular Formula

– C29H20Cl2N6O3S

References

– [1]Wen X, Zhang M, Duan Z, Suo Y, Lu W, Jin R, Mu B, Li K, Zhang X, Meng L, Hong Y, Wang X, Hu H, Zhu J, Song W, Shen A, Lu X. Discovery, SAR Study of GST Inhibitors from a Novel Quinazolin-4(1H)-one Focused DNA-Encoded Library. J Med Chem. 2023 Aug 24;66(16):11118-11132.

Molecular Weight

– 603.48

SMILES

– O=C(C1=CC(C2=C(C=CC=C2)C3=NN=NN3)=CC=C1N=C4C5=CC=C(S5)Cl)N4CC(C(O)=O)CC6=CC=C(C=C6)Cl

Clinical Information

– No Development Reported

Research Area

– others

Solubility

– 10 mM in DMSO

Target

– Gutathione S-transferase

Pathway

– Metabolic Enzyme/Protease

Product type

– Reference compound

Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.

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