Download Files:
GR125487 (sulfamate)
$417 – $667
Products Details
Product Description
– GR125487 sulfamate is an orally active and selective antagonist of 5-HT4R. GR125487 sulfamate effectively blocks the cognition enhancing effect. GR125487 sulfamate can be used to study memory disorders, gastrointestinal disorders, mood disorders and urinary tract dysfunction[1].
Web ID
– HY-103146
Shipping
– Room temperature
Molecular Formula
– C19H29FN4O8S2
References
– [1]Nirogi, R., et al. Synthesis of GR 125487, a selective 5-HT4receptor antagonist. Synthetic Communications, 46(12), 1036–1043.
CAS Number
– 859502-43-5
Molecular Weight
– 524.58
SMILES
– O=C(C1=C(NC2=C1C=C(F)C=C2)OC)OCC3CCN(CC3)CCNS(=O)(C)=O.O=S(O)(N)=O
Clinical Information
– No Development Reported
Research Area
– Neurological Disease
Solubility
– 10 mM in DMSO
Target
– 5-HT Receptor
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
