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Products Details
Product Description
– GR 89696 free base is a highly selective κ2 opioid receptor agonist with potential to prevent pruritus[1].
Web ID
– HY-107747A
Shipping
– Room temperature
Molecular Formula
– C19H25Cl2N3O3
References
– [1]Mei-Chuan Ko, et al. Effects of atypical kappa-opioid receptor agonists on intrathecal morphine-induced itch and analgesia in primates. J Pharmacol Exp Ther. 2009 Jan;328(1):193-200. |[2]A Barber, et al. Effects of GR-89696 and the novel peripherally selective OP2 agonists, EMD-61569 and EMD-61747, against focal cerebral ischemia in the rat. Methods Find Exp Clin Pharmacol. 1999 Mar;21(2):105-13
CAS Number
– 126766-31-2
Molecular Weight
– 414.33
SMILES
– O=C(N1CCN(C(CN2CCCC2)C1)C(CC3=CC=C(C(Cl)=C3)Cl)=O)OC
Clinical Information
– No Development Reported
Research Area
– Inflammation/Immunology
Solubility
– 10 mM in DMSO
Target
– Opioid Receptor
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
