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Products Details
Product Description
– GR 128107 is a competitive melatonin receptor antagonist (pKi: 9.6)[1].
Web ID
– HY-120182
Shipping
– Room temperature
Molecular Formula
– C16H20N2O2
References
– [1]Dubocovich ML, et al. Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroreceptor. Naunyn Schmiedebergs Arch Pharmacol. 1997 Mar;355(3):365-75.
CAS Number
– 190328-44-0
Molecular Weight
– 272.34
SMILES
– CC(N1CC(CCC1)C2=CNC3=C2C=C(C=C3)OC)=O
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Melatonin Receptor
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
