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GPR109 receptor agonist-1
$50 – $250
Products Details
Product Description
– GPR109 receptor agonist-1 (Compound 3a) is a highly selective agonist of the human orphan G-protein-coupled receptor GPR109b, with the pEC50 of 6.4. GPR109 receptor agonist-1 can be used for the research of cardio-metabolic diseases[1].
Web ID
– HY-107580
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Metabolism-protein/nucleotide metabolism
Molecular Formula
– C10H11N3O2
References
– [1]Graeme Semple, et al. 1-Alkyl-benzotriazole-5-carboxylic acids are highly selective agonists of the human orphan G-protein-coupled receptor GPR109b. J Med Chem. 2006 Feb 23;49(4):1227-30.
CAS Number
– 306935-41-1
Molecular Weight
– 205.21
Compound Purity
– 99.91
SMILES
– O=C(C1=CC=C(N(C(C)C)N=N2)C2=C1)O
Clinical Information
– No Development Reported
Research Area
– Cardiovascular Disease; Metabolic Disease
Solubility
– DMSO : 100 mg/mL (ultrasonic)
Target
– GPR109A
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
