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Products Details
Product Description
– GPBAR1-IN-3 (Compound 14) is a selective GPBAR1 agonist (EC50=0.17 μM) and a CysLT1R antagonist[1].
Web ID
– HY-145234
Shipping
– Room temperature
Applications
– Neuroscience-Neuromodulation
Molecular Formula
– C21H23NO2
References
– [1]Fiorillo B, et al. Structural Basis for Developing Multitarget Compounds Acting on Cysteinyl Leukotriene Receptor 1 and G-Protein-Coupled Bile Acid Receptor 1. J Med Chem. 2021 Nov 12.
CAS Number
– 2760546-05-0
Molecular Weight
– 321.41
SMILES
– CC(CC)COC1=CC(OCC2=NC3=C(C=C2)C=CC=C3)=CC=C1
Clinical Information
– No Development Reported
Research Area
– Neurological Disease; Others
Solubility
– 10 mM in DMSO
Target
– G protein-coupled Bile Acid Receptor 1;Leukotriene Receptor
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
