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Products Details
Product Description
– Glucokinase activator 1 is a liver-directed glucokinase activator with an EC50 of 34 nM.
Web ID
– HY-101788
Shipping
– Room temperature
Applications
– Metabolism-sugar/lipid metabolism
Molecular Formula
– C27H20F2N2O7S2
References
– [1]Deshpande AM, et al. Discovery of liver-directed glucokinase activator having anti-hyperglycemic effect without hypoglycemia. Eur J Med Chem. 2017 Jun 16;133:268-286.
CAS Number
– 1328987-85-4
Molecular Weight
– 586.58
SMILES
– O=S(C1=CC=C([C@H](C(NC2=NC=C(OC3=CC=C(C(O)=O)C=C3)S2)=O)OC4=CC=C(F)C=C4F)C=C1)(C5CC5)=O
Clinical Information
– No Development Reported
Research Area
– Metabolic Disease
Solubility
– 10 mM in DMSO
Target
– Glucokinase
Pathway
– Metabolic Enzyme/Protease
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
