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G244-LM
SKU
HY-117705-10 mg
Category Reference compound
Tags Cancer, Cell Cycle/DNA Damage;Epigenetics, PARP
$130 – $820
Products Details
Product Description
– G244-LM is a potent and specific inhibitor of tankyrase 1/2 that inhibits Wnt signaling[1].
Web ID
– HY-117705
Storage Temperature
– 4°C (Powder, protect from light)
Shipping
– Room Temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C18H22N4O3S2
References
– [1]Lau T, et al. A novel tankyrase small-molecule inhibitor suppresses APC mutation-driven colorectal tumor growth. Cancer Res. 2013 May 15;73(10):3132-44.
CAS Number
– 1563007-08-8
Molecular Weight
– 406.52
Compound Purity
– 98.88
SMILES
– O=C1C(CSCC2)=C2N=C(N3CCN(C4=CC=CC=C4S(=O)(C)=O)CC3)N1
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– DMSO : 6.25 mg/mL (ultrasonic;warming;heat to 80°C)
Target
– PARP
Pathway
– Cell Cycle/DNA Damage;Epigenetics
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.