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Fedovapagon
SKU
HY-14887-10 mg
Category Reference compound
Tags GPCR/G Protein, Metabolic Disease, Vasopressin Receptor
$140 – $850
Products Details
Product Description
– Fedovapagon (VA106483) is a selective and orally active vasopressin V2 receptor (V2R) agonist with an EC50 of 24 nM. Fedovapagon can be used in the research of nocturia[1].
Web ID
– HY-14887
Storage Temperature
– 4°C (Powder, stored under nitrogen)
Shipping
– Room Temperature
Applications
– Neuroscience-Neuromodulation
Molecular Formula
– C27H34N4O3
References
– [1]Yea CM, et al. New benzylureas as a novel series of potent, nonpeptidic vasopressin V2 receptor agonists. J Med Chem. 2008 Dec 25;51(24):8124-34.
CAS Number
– 347887-36-9
Molecular Weight
– 462.58
Compound Purity
– 99.14
SMILES
– CC1=C(CNC(N2CCC[C@]2(C(N(C)C)=O)[H])=O)C=CC(C(N3CCCCC4=C3C=CC=C4)=O)=C1
Clinical Information
– Phase 3
Research Area
– Metabolic Disease
Solubility
– DMSO : ≥ 125 mg/mL
Target
– Vasopressin Receptor
Isoform
– V2 ReceptorÂ
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.