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Products Details
Product Description
– FAP-IN-1 is a fibroblast activation protein (FAP) inhibitor with an IC50 value of 3.3 nM. FAP-IN-1 can be used for the research of cancer[1].
Web ID
– HY-149860
Shipping
– Room temperature
Molecular Formula
– C65H88F2N12O18
References
– [1]Wang Y, et al. High Affinity and FAP-Targeted Radiotracers: A Potential Design Strategy to Improve the Pharmacokinetics and Tumor Uptake for FAP Inhibitors. J Med Chem. 2023 Jul 13;66(13):8614-8627.
Molecular Weight
– 1363.46
SMILES
– O=C(C1=CC=NC2=C1C=CC=C2NC([C@H](CCCCNC(CCOCCOCCOCCOCCOCCOCCNC(CN3CCN(CCN(CCN(CC3)CC(O)=O)CC(O)=O)CC(O)=O)=O)=O)NC(C4=C5C=CC=CC5=CC=C4)=O)=O)NCC(N6[C@@](C#N)(CC(F)(C6)F)[H])=O
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– FAP
Pathway
– Immunology/Inflammation
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
