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Products Details
Product Description
– Estrogen receptor β antagonist 2 is a potent and selective estrogen receptor β (ERβ) antagonist with IC50s of 109.10, 0.63 µM for Erα and Erβ, respectively[1].
Web ID
– HY-150693
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C23H26N2O6
References
– [1]Carr M, et al. Optimisation of estrogen receptor subtype-selectivity of a 4-Aryl-4H-chromene scaffold previously identified by virtual screening. Bioorg Med Chem. 2020 Mar 1;28(5):115261.
CAS Number
– 2580941-14-4
Molecular Weight
– 426.46
SMILES
– O=C(C1=C(N)OC2=C(C=CC(O)=C2)C1C3=CC=C(OCCN4CCOCC4)C=C3)OC
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Estrogen Receptor/ERR
Isoform
– ERα;ERβ
Pathway
– Vitamin D Related/Nuclear Receptor
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
