Download Files:
Eprazinone (dihydrochloride)
SKU
HY-B2078A-100 mg
Category Reference compound
Tags GPCR/G Protein;Neuronal Signaling, Inflammation/Immunology, Neurokinin Receptor
$40 – $210
Products Details
Product Description
– Eprazinone dihydrochloride is a gent with mucolytic, secretolytic, antitussive, and bronchial antispasmodic properties. Eprazinone dihydrochloride is a neurokinin 1 receptor (NK1R) ligand. Eprazinone dihydrochloride has the potential for chronic bronchitis treatment that improved pulmonary function and arterial partial pressure of oxygen[1][2].
Web ID
– HY-B2078A
Storage Temperature
– 4°C (Powder, sealed storage, away from moisture)
Shipping
– Room Temperature
Applications
– COVID-19-immunoregulation
Molecular Formula
– C24H34Cl2N2O2
References
– [1]R S Thrall, et al. Eprazinone Alters Lung Lavage Lipid Levels and Transtracheal Ion Transport. Exp Lung Res. May-Jun 1992;18(3):409-20.|[2]Yvonne Krautscheid, et al. Pharmacophore Modeling, Virtual Screening, and in Vitro Testing Reveal Haloperidol, Eprazinone, and Fenbutrazate as Neurokinin Receptors Ligands. J Chem Inf Model. 2014 Jun 23;54(6):1747-57.
CAS Number
– 10402-53-6
Molecular Weight
– 453.44
Compound Purity
– 98.0
SMILES
– O=C(C1=CC=CC=C1)C(C)CN2CCN(CC(OCC)C3=CC=CC=C3)CC2.Cl[H].Cl[H]
Clinical Information
– Launched
Research Area
– Inflammation/Immunology
Solubility
– DMSO : 6.25 mg/mL (ultrasonic;warming;heat to 60°C)|H2O : ≥ 25 mg/mL
Target
– Neurokinin Receptor
Isoform
– NK1
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.