Download Files:
EP3 antagonist 3
$300 – $2,400
Products Details
Product Description
– EP3 antagonist 3 (compound 2) is an orally active, potent and selective EP3 antagonist, with a pKi of 8.3. EP3 antagonist 3 shows excellent pharmacokinetic properties. EP3 antagonist 3 can be used for overactive bladder (OAB) research[1].
Web ID
– HY-147226
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Metabolism-protein/nucleotide metabolism
Molecular Formula
– C21H18N2O4
References
– [1]Jin J, et al. Novel 3-Oxazolidinedione-6-aryl-pyridinones as Potent, Selective, and Orally Active EP3 Receptor Antagonists. ACS Med Chem Lett. 2010 May 14;1(7):316-20.
CAS Number
– 1227827-88-4
Molecular Weight
– 362.38
Compound Purity
– 99.57
SMILES
– O=C1OC(C2=CC=C(C3=CC4=C(C=CC=C4)C=C3)NC2=O)(C(C)C)C(N1)=O
Clinical Information
– No Development Reported
Research Area
– Endocrinology; Neurological Disease
Solubility
– DMSO : 250 mg/mL (ultrasonic)
Target
– Prostaglandin Receptor
Isoform
– EP
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
