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EP1-antagonist-1
$315
Only 1000 item(s) left in stock.
Products Details
Product Description
– EP1-antagonist-1 is a EP1 antagonist with a pKi of 7.54 and an pIC50 of 8.5[1].
Web ID
– HY-101695
Shipping
– Room temperature
Applications
– Metabolism-protein/nucleotide metabolism
Molecular Formula
– C19H15BrCl2N2O3
References
– [1]McKeown SC, et al. Identification of novel pyrazole acid antagonists for the EP1 receptor. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4767-71. Epub 2006 Jul 14.
CAS Number
– 851204-35-8
Molecular Weight
– 470.14
SMILES
– O=C(C1=NN(CC2=CC(Br)=CC=C2OCC3=CC=C(Cl)C=C3Cl)C(C)=C1)O
Clinical Information
– No Development Reported
Research Area
– Neurological Disease; Endocrinology
Solubility
– 10 mM in DMSO
Target
– Prostaglandin Receptor
Isoform
– EP
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
