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Products Details
Product Description
– Enofelast (BI-L-239), a 5-lipoxygenase (5-LO) inhibitor, exhibits an IC50 of 2.48 μM for inhibition of calcium ionophore-induced LTB4 generation[1].
Web ID
– HY-120539
Shipping
– Room temperature
Molecular Formula
– C16H15FO
References
– [1]T C Noonan, et al. Effect of BI-L-239, A-64077 and MK-886 on leukotriene B4 synthesis by chopped guinea pig lung and on antigen-induced tracheal contraction in vitro. Prostaglandins. 1992 Dec;44(6):543-54.
CAS Number
– 125722-16-9
Molecular Weight
– 242.29
SMILES
– OC1=C(C=C(C=C1C)/C=C/C2=CC=C(C=C2)F)C
Clinical Information
– No Development Reported
Research Area
– Inflammation/Immunology
Solubility
– 10 mM in DMSO
Target
– Leukotriene Receptor;Lipoxygenase
Pathway
– GPCR/G Protein;Metabolic Enzyme/Protease
Product type
– Reference compound
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