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Products Details
Product Description
– ENMD-1068 hydrobromide is a potent PAR2 antagonist. ENMD-1068 hydrobromide attenuates joint inflammation in a dose-dependent manner. ENMD-1068 hydrobromide can be used in research of joint inflammation[1].
Web ID
– HY-122049
Shipping
– Room temperature
Applications
– COVID-19-immunoregulation
Molecular Formula
– C15H30BrN3O2
References
– [1]Kelso EB, et, al. Therapeutic promise of proteinase-activated receptor-2 antagonism in joint inflammation. J Pharmacol Exp Ther. 2006 Mar;316(3):1017-24.
CAS Number
– 644961-61-5
Molecular Weight
– 364.32
SMILES
– O=C(N1CCN(C(CC(C)C)=O)CC1)CCCCCN.Br
Clinical Information
– No Development Reported
Research Area
– Inflammation/Immunology
Solubility
– 10 mM in DMSO
Target
– Protease Activated Receptor (PAR)
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
