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Empesertib
SKU
HY-12858-10 mg
Category Reference compound
Tags Cancer, Cell Cycle/DNA Damage;Cytoskeleton, Mps1
$290 – $2,520
Products Details
Product Description
– Empesertib (BAY 1161909) is a potent Mps1 inhibitor, with an IC50 of < 1 nM.
Web ID
– HY-12858
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C29H26FN5O4S
References
– [1]SCHULZE, Volker, et al. PRODRUG DERIVATIVES OF SUBSTITUTED TRIAZOLOPYRIDINES. WO2014198647A2
CAS Number
– 1443763-60-7
Molecular Weight
– 559.61
Compound Purity
– 98.82
SMILES
– FC1=CC=C([C@@H](C)C(NC2=CC=C(C3=CN4N=C(NC5=CC=C(S(C)(=O)=O)C=C5OC)N=C4C=C3)C=C2)=O)C=C1
Clinical Information
– Phase 1
Research Area
– Cancer
Solubility
– DMSO : ≥ 35 mg/mL
Target
– Mps1
Pathway
– Cell Cycle/DNA Damage;Cytoskeleton
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.