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E1R
$307 – $2,250
Products Details
Product Description
– E1R is a positive allosteric modulator of sigma-1 receptors (Sig1R PAM) with cognition-enhancing activity[1].
Web ID
– HY-116463
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Neuroscience-Neuromodulation
Molecular Formula
– C13H16N2O2
References
– [1]Zvejniece L, et al. The cognition-enhancing activity of E1R, a novel positive allosteric modulator of sigma-1 receptors. Br J Pharmacol. 2014 Feb;171(3):761-71.
CAS Number
– 1301211-78-8
Molecular Weight
– 232.28
Compound Purity
– 99.28
SMILES
– O=C(CN1C(C[C@@H]([C@@H]1C)C2=CC=CC=C2)=O)N
Clinical Information
– No Development Reported
Research Area
– Neurological Disease
Solubility
– DMSO : 60 mg/mL (ultrasonic)
Target
– Sigma Receptor
Isoform
– Sigma 1 Receptor
Pathway
– Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
