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Didesmethyl cariprazine

SKU HY-100658-10 mg Category Reference compound Tags 5-HT Receptor;Dopamine Receptor, GPCR/G Protein;Neuronal Signaling, Neurological Disease

$550 – $2,820

Size10 mg

5 mg 10mM/1mL 10 mg 25 mg 50 mg

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$880

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Products Details

Product Description

– Didesmethyl cariprazine is a metabolite of Cariprazine and acts as the predominant circulating active moiety. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a antipsychotic agent candidate that exhibits high affinity for the D3 and D2 receptors, and moderate affinity for the 5-HT1A receptor[1].

Web ID

– HY-100658

Storage Temperature

– -20°C, 3 years; 4°C, 2 years (Powder)

Shipping

– Room Temperature

Applications

– Neuroscience-Neuromodulation

Molecular Formula

– C19H28Cl2N4O

References

– [1]Citrome L, et al. Cariprazine for acute and maintenance treatment of adults with schizophrenia: an evidence-based review and place in therapy. Neuropsychiatr Dis Treat. 2018 Oct 5;14:2563-2577.

CAS Number

– 839712-25-3

Molecular Weight

– 399.36

Compound Purity

– 99.79

SMILES

– O=C(N)N[C@H]1CC[C@H](CCN2CCN(C3=CC=CC(Cl)=C3Cl)CC2)CC1

Clinical Information

– No Development Reported

Research Area

– Neurological Disease

Solubility

– DMSO : 11.36 mg/mL (ultrasonic;warming;heat to 80°C)

Target

– 5-HT Receptor;Dopamine Receptor

Isoform

– 5-HT1 Receptor;D2 Receptor;D3 Receptor

Pathway

– GPCR/G Protein;Neuronal Signaling

Product type

– Reference compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.