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Products Details
Product Description
– Debrisoquin (Isocaramidine) is a TMPRSS2 inhibitors that inhibits SARS-CoV-2 entry into human lung cell line by a TMPRSS2-depedent manner, with an IC50 of 22μM. Debrisoquin can be used for antiviral research[1].
Web ID
– HY-B1624
Shipping
– Room temperature
Molecular Formula
– C10H13N3
References
– [1]Amanda L. Peiffer, et.al.TMPRSS2 Inhibitor Discovery Facilitated through an In Silico and Biochemical Screening Platform.ACS Medicinal Chemistry Letters 2023 14 (6), 860-866.
CAS Number
– 1131-64-2
Molecular Weight
– 175.23
SMILES
– NC(N1CCC2=C(C1)C=CC=C2)=N
Clinical Information
– No Development Reported
Research Area
– Infection
Solubility
– 10 mM in DMSO
Target
– SARS-CoV;Ser/Thr Protease
Isoform
– Human Endogenous Metabolite
Pathway
– Anti-infection;Metabolic Enzyme/Protease
Product type
– Natural Products
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