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Cyclobenzaprine-d3 (hydrochloride)
SKU
HY-B0740S-1 mg
Category Isotope-Labeled Compounds
Tags 5-HT Receptor;Isotope-Labeled Compounds, GPCR/G Protein;Neuronal Signaling;Others, Neurological Disease
Products Details
Product Description
– Cyclobenzaprine-d3 (hydrochloride) is the deuterium labeled Cyclobenzaprine hydrochloride. Cyclobenzaprine hydrochloride (MK130 hydrochloride) is a skeletal muscle relaxant and a central nervous system (CNS) depressant.
Web ID
– HY-B0740S
Shipping
– Room temperature
Molecular Formula
– C20H19D3ClN
References
– [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216. |[2]Kobayashi, H., Y. Hasegawa, and H. Ono, Cyclobenzaprine, a centrally acting muscle relaxant, acts on descending serotonergic systems. Eur J Pharmacol, 1996. 311(1): p. 29-35.|[3]Honda, M., T. Nishida, and H. Ono, Tricyclic analogs cyclobenzaprine, amitriptyline and cyproheptadine inhibit the spinal reflex transmission through 5-HT(2) receptors. Eur J Pharmacol, 2003. 458(1-2): p. 91-9.
CAS Number
– 1184983-42-3
Molecular Weight
– 314.87
SMILES
– [2H]C([2H])([2H])N(C)CC/C=C1C2=CC=CC=C2C=CC3=CC=CC=C13.Cl
Clinical Information
– No Development Reported
Research Area
– Neurological Disease
Solubility
– 10 mM in DMSO
Target
– 5-HT Receptor;Isotope-Labeled Compounds
Pathway
– GPCR/G Protein;Neuronal Signaling;Others
Product type
– Isotope-Labeled Compounds
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