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Products Details
Product Description
– Ceefourin 2 is a potent and highly selective inhibitor of MRP4. Ceefourin 2 inhibits the transport of MRP4 substrates but is not selective for other ABC transporters. Ceefourin 2 shows lower cytotoxicity and higher microsomal and acid stability[1].
Web ID
– HY-121088
Shipping
– Room temperature
Molecular Formula
– C15H9ClF3N3O2
References
– [1]Cheung L, et al. High-throughput screening identifies Ceefourin 1 and Ceefourin 2 as highly selective inhibitors of multidrug resistance protein 4 (MRP4). Biochem Pharmacol. 2014 Sep 1;91(1):97-108.
CAS Number
– 348148-51-6
Molecular Weight
– 355.70
SMILES
– O=C(O)C1=NN2C(C(F)(F)F)=CC(C3=CC=C(C=C3)C)=NC2=C1Cl
Clinical Information
– No Development Reported
Research Area
– Cardiovascular Disease; Others
Solubility
– 10 mM in DMSO
Target
– Others
Pathway
– Others
Product type
– Reference compound
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