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CDK9-IN-8
$350 – $2,250
Products Details
Product Description
– CDK9-IN-8 is a highly effective and selective CDK9 inhibitor with an IC50 of 12 nM.
Web ID
– HY-102039
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Cancer-Kinase/protease
Molecular Formula
– C31H32FN7O3
References
– [1]Li Y, et al. Discovery of a highly potent, selective and novel CDK9 inhibitor as an anticancer drug candidate. Bioorg Med Chem Lett. 2017 Aug 1;27(15):3231-3237.
CAS Number
– 2105956-51-0
Molecular Weight
– 569.63
Compound Purity
– 99.65
SMILES
– FC1=CC=C(NC(C2(CC2)C(NC3=CC=C(NC4=NC=C5C(N(C6CCCC6)C(C(N(C)C)=O)=C5)=N4)C=C3)=O)=O)C=C1
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– DMSO : 5.2 mg/mL (ultrasonic;warming;heat to 80°C)|H2O : 1 mg/mL (ultrasonic;warming;heat to 80°C)
Target
– CDK
Isoform
– CDK9
Pathway
– Cell Cycle/DNA Damage
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
