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Products Details
Product Description
– CBK289001 is a tartrate-resistant acid phosphatase (TRAP/ACP5) inhibitor. CBK289001 inhibits TRAP 5bMV, TRAP 5bOX and TRAP 5aOX with IC50s of 125 µM, 4.21 µM and 14.2 µM, respectively[1].
Web ID
– HY-124663
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C19H20N6O4
References
– [1]Anja Reithmeier, et al. Identification of inhibitors of Tartrate-resistant acid phosphatase (TRAP/ACP5) activity by small-molecule screening. Chem Biol Drug Des. 2018 Jul;92(1):1255-1271.
CAS Number
– 1212663-24-5
Molecular Weight
– 396.40
SMILES
– O=C(N1[C@H](C2=NC(C3=CC=C(OCO4)C4=C3)=NO2)CC5=C(NC=N5)C1)NC(C)C
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Protease Activated Receptor (PAR)
Pathway
– GPCR/G Protein
Product type
– Reference compound
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