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Products Details
Product Description
– CB2 receptor antagonist 3 (compound (S)-1) is an inverse agonist of the cannabinoid receptor CB2R with Kd=39 nM. CB2 receptor antagonist 3 can be used as a tool to synthesize a variety of CB2R probes[1].
Web ID
– HY-155481
Shipping
– Room temperature
Molecular Formula
– C33H46N4O2
References
– [1]Carreira E et al. Flipping the GPCR Switch: Structure–Based Development of Selective Cannabinoid Receptor 2 Inverse Agonists[J]. 2023.
Molecular Weight
– 530.74
SMILES
– CC(C1=CC(OC)=C([C@@]2([H])C=C(CN)[C@@H]3C(C)(C)[C@H]2C3)C(OC)=C1)(C)[C@@H](CCCCCN=[N+]=[N-])C4=CC=CC=C4
Clinical Information
– No Development Reported
Research Area
– Neurological Disease
Solubility
– 10 mM in DMSO
Target
– Cannabinoid Receptor
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
