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Products Details
Product Description
– CB1 inverse agonist 2 is an orally active inverse agonist of Cannabinoid Receptor CB1. CB1 inverse agonist 2 effectively inhibits CP55940-induced hypothermia and anorexia in mice model[1].
Web ID
– HY-12095
Shipping
– Room temperature
Molecular Formula
– C24H20ClFN2OS
References
– [1]Synthesis and Evaluation of Dibenzothiazepines: A Novel Class of Selective Cannabinoid-1 Receptor Inverse Agonists
J. Med. Chem., 2009, 52 (7), pp 1975-1982|[2]Pettersson H, et al. Synthesis and evaluation of dibenzothiazepines: a novel class of selective cannabinoid-1 receptor inverse agonists. J Med Chem. 2009 Apr 9;52(7):1975-82.
CAS Number
– 1019839-52-1
Molecular Weight
– 438.94
SMILES
– O=C(C1=CC=C2SC3=CC=CC=C3C(C4=CC=C(F)C(Cl)=C4)=NC2=C1)NCCCC
Clinical Information
– No Development Reported
Research Area
– Neurological Disease
Solubility
– 10 mM in DMSO
Target
– Cannabinoid Receptor
Isoform
– CB1;CB2
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
