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Products Details
Product Description
– CARM1-IN-3 (compound 17b) is a potent and selective co-activator associated arginine methyltransferase (CARM1) inhibitor with IC50 values of 0.07, >25 µM for CARM1 and CARM3, respectively[1].
Web ID
– HY-15214
Shipping
– Room temperature
Molecular Formula
– C24H32N4O2
References
– [1]Wan H, et al. Benzo[d]imidazole inhibitors of Coactivator Associated Arginine Methyltransferase 1 (CARM1)–Hit to Lead studies. Bioorg Med Chem Lett. 2009 Sep 1;19(17):5063-6.
CAS Number
– 912970-67-3
Molecular Weight
– 408.54
SMILES
– CNCCN1CCC(C2=CC3=C(N=C(C4=C(OC)C=CC=C4OC)N3)C(C)=C2)CC1
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Histone Methyltransferase
Pathway
– Epigenetics
Product type
– Reference compound
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