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Calpain-2-IN-1
$480 – $4,200
Products Details
Product Description
– Calpain-2-IN-1 (Formula 1A) is a isoform-specific calpain-2 inhibitor with Kis of 181 nM and 7.8 nM for calpain-1, and calpain-2, respectively. Calpain-2-IN-1 can be used for the research of neurodegenerative diseases and other diseases of synaptic function[1].
Web ID
– HY-145155
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Metabolism-protein/nucleotide metabolism
Molecular Formula
– C28H37N3O7
References
– [1]Michel Baudry, et al. Isoform-specific calpain inhibitors, methods of identification, and uses thereof. WO2016077461A2.
CAS Number
– 144231-85-6
Molecular Weight
– 527.61
Compound Purity
– 98.84
SMILES
– O=C(OCC1=CC=CC=C1)N[C@@H](CC(C)C)C(N[C@@H](CC)C(C(NCC2=CC(OC)=CC(OC)=C2)=O)=O)=O
Clinical Information
– No Development Reported
Research Area
– Neurological Disease
Solubility
– DMSO : 100 mg/mL (ultrasonic)
Target
– Proteasome
Pathway
– Metabolic Enzyme/Protease
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
