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Products Details
Product Description
– c-Myc inhibitor 5 (DA3) is a fluorescent, long chain-bridged bispurine that selectively targets the c-MYC G-quadruplex (KD of 16 μM). c-Myc inhibitor 5 shows inhibition on c-MYC expression rather than other G4-driven oncogenes[1].
Web ID
– HY-145843
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C30H46N12
References
– [1]Hu MH, et al. Discovery of a fluorescent, long chain-bridged bispurine that selectively targets the c-MYC G-quadruplex. Bioorg Chem. 2022;122:105750.
Molecular Weight
– 574.77
SMILES
– CC1CCN(CC1)C2=NC(N)=C3N=CN(C3=N2)CCCCCCCCN4C5=NC(N6CCC(C)CC6)=NC(N)=C5N=C4
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– c-Myc
Pathway
– Apoptosis
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
