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BRD4-BD1/2-IN-2
SKU
HY-142675-Get quote
Category Reference compound
Tags Cancer, Epigenetic Reader Domain, Epigenetics
Products Details
Product Description
– BRD4-BD1/2-IN-2 is a potent BRD4 BD2 inhibitor with IC50s of <0.5 nM and <300 nM for BRD4 BD2 and BRD4 BD1, respectively (WO2021233371A1, compound 2)[1].
Web ID
– HY-142675
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C30H33N5O4
References
– [1]Compound functioning as bromodomain protein inhibitor, and composition. WO2021233371A1.
CAS Number
– 2743464-27-7
Molecular Weight
– 527.61
SMILES
– O=C(C1=CC(C(C2=CC3=NN(CC(C)(C)O)C=C3C=C2OC4=C(C)C=CC=C4C)=CN5C)=C(N1)C5=O)NCC
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Epigenetic Reader Domain
Pathway
– Epigenetics
Product type
– Reference compound
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